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Pharmacology · CNS drugs
Sample itemWhich receptor complex is enhanced by benzodiazepines to increase inhibitory signaling?
Original practice item, not a recalled exam question. Nothing here is recorded.
The answer and the reasoning
D. GABA-A receptor
Benzodiazepines enhance GABA-A receptor activity by increasing the frequency of chloride-channel opening, producing anxiolytic, sedative, anticonvulsant, and muscle-relaxant effects.
Option by option
A. NMDA receptor
NMDA receptor activity is not the primary benzodiazepine target.
B. Dopamine D2 receptor
D2 receptors are targeted by many antipsychotics.
C. Beta-1 receptor
Beta-1 receptors are cardiac adrenergic receptors.
D. GABA-A receptor (correct)
Correct: benzodiazepines enhance GABA-A mediated inhibition.
Source note: Original NextPrep sample item — pending expert review. This item is original practice material awaiting independent expert review, so confirm important facts in a standard textbook.